A short review on sulphonamides with antimicrobial activity
DOI:
https://doi.org/10.7439/ijpc.v7i5.4125Keywords:
chromosomal Abnormality, Spontaneous Abortion, aneuploidyAbstract
Sulfonamides are one of the organosulphur compounds containing the -SO2NH2 and/or -SO2NH- group(s). The sulphonamides or sulfa drugs competitively inhibit folic acid synthesis in micro-organisms and subsequently inhibit multiplication of bacteria but do not actively kill them. They have been used against most gram-positive and many gram-negative bacteria, some fungi, and certain protozoa. Medically important sulphonamidesDownloads
References
Siddique Muddassar, Saeed B. A., Ahmad S., Dogar A. N., Synthesis and Biological Evaluation of Hydrazide based Sulfonamides, Journal of Scientific & Innovative Research, 2013, vol.2, Issue 3, pp. 627-633.
Al-Mudhafar Jawad May Mohammed, Abdulkadir Qusay Maadh, Mohammed Abbas Amera, Hussian Mohammed Azhar, A Al-hilli Faris , Synthesis and Microbiological Study Of New Sulfonamide , International Journal Of Comprehensive Pharmacy Research, 2012, vol.6, Issue 2, pp. 976-8157.
Santosh, Kumar; Niranjan M S, Chaluvaraju, K C; Jamakhandi, C M;Dayanand, Kadadevar, 2010,Synthesis and Antimicrobial Study of Some Schiff Bases of Sulfonamides Journal of Current Pharmaceutical Research,vol.01 pp. 39-42
Gleckman R, Alvarez S, Joubert DW; Drug therapy reviews: trimethoprim-sulfamethoxazole. Am J Hosp Pharm. 1979; vol 36, Issue 7, pp. 893-906.
Hossein Eshghia, Mohammad Rahimizadeh, MahmoodZokaei, Shaghayegh Eshghi, Shohreh Eshghi, ZinaFaghihi, Elaheh Tabasi and Mehdi Kihanyan; Synthesisand antimicrobial activity of some new macrocyclicbis- sulfonamide and disulfides, European Journal of Chemistry. 2011; vol 2 Issue1, pp 47-50.
Fujita T., Hansch C.: (1967); Analysis of the Structure-Activity Relationship of the Sulfonamide Drugs Using Substituent Constants. J.Med.Chem. vol.10 pp.991.
Anand N, (1996); Sulfonamides and Sulfons. In Wolff M E (ed.). Burger
Eshghia H., Rahimizadeh M., Zokaei M., Eshghi S., Eshghi S., Faghihi Z., Tabasi Z. Kihanyan M.:(2011);Synthesis and antimicrobial activity of some new macrocyclic
Locuson, C. W.; Gannett, P. M.; Ayscue, R.; Tracy, T. S. Use of simple docking methods to screen a virtual library for heteroactivators of cytochrome P450 2C9. J. Med. Chem., 50(6):1158- 1165,(2007)
Boison, J. O.; Nachilobe, P.; Cassidy, R.; Keng, L.; Thacker, P. A.; Peacock, A.; Fesser, A. C.; Lee, S.; Korsrud, G. O.; Bulmer, W. S. Determination of trimethoprim and sulphadoxine residues in porcine tissues and plasma. Canadian J. Vet. Res., 60(4):281-287,(1996)
Rosen B. R., Ruble J. C., Beauchamp T. J., Navarro A.:( 2011); Mild Pd-Catalyzed N-Arylation of Methanesulfonamide and Related Nucleophiles: Avoiding Potentially Genotoxic Reagents and Byproducts. Org. Lett.vol,13,pp. 2564
Dogruer, D. S.; Urlu, S.; Onkol, T.; Ozcellik, B.; Sahin, M. F.(2010) Synthesis of some pyridazine derivatives carrying urea, thiourea,and sulfonamide moieties and their antimicrobial activity. Turkey J. Chem., Vol,34pp:.57-65 .
Veisi H.,Ghorbani-Vaghei R.,Hemmati S., Mahmoodi J.: (2011);Convenient One-Pot Synthesis of Sulfonamides and Sulfonyl Azides from Thiols Using N-Chlorosuccinimide. Synlett, vol, 16,pp. 2315.
Jiao, Z.-G.; He, H.-Q.; Zeng, C.-C.; Tan, J.-J.; Hu, L.-M.; Wang, C.-X.( 2010,Design, synthesis and anti-HIV integrase evaluation of N-(5-chloro-8-hydroxy-2- styrylquinoline-7-yl) benzenesulfonamide derivatives. Molecules, vol,15(3)pp.1903-1917
Y Genc, R Ozkanca, Y Bekdemir. Ann Clin Microb Antimicrob 2008, 7-17
:17doi:10:1186/1476-0711.
Iro, Argyropoulou;a Athina, Geronikaki; Paola, Vicini; Franca, Zanib; 2009 Synthesis and biological evaluation of sulfonamide thiazole and benzothiazole derivatives as antimicrobial agents, ARKIVOCVOL,(vi)PP. 89-102
HUSAIN, ASIF; 2009.Amide Derivatives of sulfonamide and isoniazid: synthesis And biological evaluation, Acta Poloniae Pharmaceutical Drug Research, Vol. 66, pp. 513-521
T. Narasaiaha, D. Subba Raoa, K. Venkata Ramanaa, S. Adamb and C. Naga Rajua 2012, Synthesis of New Sulfonamide Derivatives of Tryptamine and TheirAntimicrobial Activity, Scholars Research Library Der Pharma Chemica,VOl, 4,Issue,(4)pp,1582-1590
Im
Abdulhakeem, Alsughaye;, Abdel-Zaher A. Elassar, Seham Mustafa1; Fakhreia; Sagheer;2011Synthesis, Structure Analysis and Antibacterial Activity of New Potent Sulfonamide DerivativesJournal of Biomaterials and Nanobiotechnology, ,Vol, 2, pp.144-149
Mostaf.M..Ghorab, Fatma A.Ragab, Helmy I. Heiba, Hebaallah M. Agha, 2011 Synthesis of Some Novel Sulfonamides ContainingBiologically Active AlkanoicAcid, Acetamide, Thiazole, and Pyrrole Moieties of Expected Antitumor andRadiosensitizing ActivitiesJ. Basic. Appl .Chem. Vol.1,Issue(2),pp.8-14,
Nadeem S., Surendra Nath P., Suroor A. K., James P. S., Arpana R., Mahfuz A. Md. Faiz A., Mashooq A., (2007)
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